Gypostemma extract is an active ingredient derived from the whole plant of the Cucurbitaceae species Gynostemma pentaphyllum, primarily produced through water extraction, alcohol extraction, or modern separation and purification techniques. Its core active compounds are gypenosides, which are structurally similar to some hits of ginsenosides, earning it the nickname "Southern Ginseng." It also contains polysaccharides, flavonoids, and other components. As a traditional medicinal and edible plant in China, Gypostemma has a long history of folk use. Modern research employs techniques like high-performance liquid chromatography to standardize the quantification of gypenosides, ensuring consistent quality and bioactivity.

Gypostemma extract exhibits a wide range of physiological regulatory functions. Its gypenosides can help regulate blood lipids and reduce blood viscosity, benefiting cardiovascular health. Its antioxidant and immune-boosting effects contribute to delaying aging and enhancing resistance. Studies have found that it can help maintain blood sugar balance through multi-target regulation of glucose metabolism. Additionally, Gypostemma extract has potential benefits such as anti-fatigue properties, improved sleep, hepatocyte protection, and inhibition of tumor cell proliferation, making it a natural extract with comprehensive regulatory effects.

Gypostemma extract is widely used in the health food industry, often as a raw material for capsules or tablets aimed at regulating blood lipids and blood sugar, as well as boosting immunity. It serves as a natural health additive in functional beverages and tea products. In pharmaceutical development, it is used in auxiliary cardiovascular and cerebrovascular treatments and liver-protecting medications. The cosmetics industry utilizes its antioxidant properties in anti-aging skincare products. In recent years, it has gained increasing attention for its applications in medical foods, sports nutrition products, and as a natural botanical ingredient in the international export market.